SCHEMBL4402972

SCHEMBL4402972

CCC(=O)c1ccc2c(OC)n[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
MAP2K4 P45985 2/20 0.40
MAPK1 P28482 10/20 0.40
KDM4E B2RXH2 1/20 0.40
ACACB O00763 1/20 0.40
ACACA Q13085 1/20 0.40
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TRPA1 O75762 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4404504 0.89 MEN1 (0.45) MEN1KMT2AMAP2K4MAPK1KDM4E
SCHEMBL30189262 0.84 MAP2K4 (0.47) MAP2K4MAPK1KDM4EACACBACACA
SCHEMBL2671667 0.84 MAP2K4 (0.47) MAP2K4MAPK1KDM4EACACBACACA
SCHEMBL25139495 0.81 ABL1 (0.51)
SCHEMBL4137466 0.80 ACACB (0.44) MAP2K4MAPK1ACACBACACARAB9A
SCHEMBL4407779 0.77 GSK3B (0.47)
SCHEMBL2300578 0.74 MAPK1 (0.42) MAPK1KDM4E
SCHEMBL2300575 0.74 MAPK1 (0.42) MAPK1KDM4E
SCHEMBL14038753 0.72 KDR (0.41) MAPK1
SCHEMBL2671776 0.72 MAP2K4 (0.50) MAP2K4MAPK1KDM4EACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed