SCHEMBL4402977

SCHEMBL4402977

CCC(=O)c1cc(C)c2[nH]nc(C)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
LMNA P02545 2/20 0.38
PPARA Q07869 2/20 0.37
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.33
PDE4D Q08499 1/20 0.33
BRD4 O60885 1/20 0.33
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ATM Q13315 1/20 0.31
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4402971 0.81 ADORA2A (0.41) ADORA2AADORA2BL3MBTL1LMNAALDH1A1
SCHEMBL30809494 0.81 ADORA2A (0.41) ADORA2AADORA2BLMNAALDH1A1KDM4E
SCHEMBL1145053 0.81 ADORA2A (0.41) ADORA2AADORA2BLMNAALDH1A1KDM4E
SCHEMBL4140051 0.77 ADORA2A (0.38) ADORA2AADORA2BLMNA
SCHEMBL4403122 0.76 MAPK1 (0.43) LMNAKDM4EMAPTATMPAK1
SCHEMBL1144961 0.73 MEN1 (0.39) ADORA2AADORA2BLMNAALDH1A1KDM4E
SCHEMBL4403674 0.73 ACACB (0.43)
SCHEMBL9720573 0.70 PPARA (0.46) L3MBTL1PPARAALDH1A1KDM4EHPGD
SCHEMBL13675149 0.70 ADORA2A (0.43) ADORA2AADORA2BLMNAALDH1A1KDM4E
SCHEMBL1144623 0.70 CA12 (0.49) ALDH1A1KDM4EHPGDCYP2C19PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed