SCHEMBL4403700

SCHEMBL4403700

CC(=O)Nc1ccc(F)c(C(=N)NO)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.49
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HDAC1 Q13547 3/20 0.44
CDK1 P06493 1/20 0.42
IDO1 P14902 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
TNNI3 P19429 1/20 0.41
TNNT2 P45379 1/20 0.41
TNNC1 P63316 1/20 0.41
RUNX1 Q01196 1/20 0.41
CBFB Q13951 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405935 0.84 SMN1; SMN2 (0.55) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL4078006 0.82 SMN1; SMN2 (0.60) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL1655468 0.80 MYC (0.56) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL2902152 0.79 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL17307570 0.76 SMN1; SMN2 (0.50) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL863069 0.76 RAB9A (0.58) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL30368269 0.76 RAB9A (0.58) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL147440 0.75 IDO1 (0.65) SMN1; SMN2MEN1KMT2AMAPTALDH1A1
SCHEMBL14100443 0.74 KAT6A (0.40) SMN1; SMN2MEN1KMT2AALDH1A1HDAC1
SCHEMBL17244480 0.73 HDAC1 (0.58) SMN1; SMN2ALDH1A1HDAC1CDK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed