SCHEMBL4408407

SCHEMBL4408407

CCc1cc(NC(=O)Cn2cc(-c3ccc(Cl)cc3)c(=O)c3ccc(C)cc32)no1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP10 Q14694 6/20 0.50
RXFP1 Q9HBX9 2/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.38
MAPK1 P28482 1/20 0.37
MAPT P10636 5/20 0.37
POLB P06746 2/20 0.37
ALDH1A1 P00352 1/20 0.36
ESR1 P03372 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4402775 0.91 USP10 (0.41) USP10RXFP1LMNAMAPK1MAPT
SCHEMBL1923430 0.90 USP10 (0.52) USP10MEN1KMT2AHSD17B10MAPK1
SCHEMBL1923423 0.84 GAPDH (0.48) USP10LMNAMEN1KMT2AHSD17B10
SCHEMBL1923540 0.81 USP10 (0.45) USP10RXFP1LMNAKMT2AMAPT
SCHEMBL1923607 0.81 CTSL (0.47) USP10LMNAMEN1KMT2AHSD17B10
SCHEMBL1923492 0.81 USP10 (0.53) USP10RXFP1LMNAMEN1KMT2A
SCHEMBL1923682 0.80 USP10 (0.49) USP10RXFP1LMNAMEN1KMT2A
SCHEMBL27775353 0.79 USP10 (0.51) USP10RXFP1LMNAMAPTPOLB
SCHEMBL1923811 0.78 USP10 (0.45) USP10LMNAMEN1KMT2AMAPT
SCHEMBL1923845 0.78 USP10 (0.48) USP10MAPTPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064185-A1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS Ferrer Internacional, S.A. (ES) 2009-06-03 EP disclosed
WO-2008017710-A1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS FERRER INTERNACIONAL S.A. (ES) 2008-02-14 WO disclosed