SCHEMBL4412970

SCHEMBL4412970

Clc1cccc(Oc2ccc3ncncc3c2)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.56
MAP4K4 O95819 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ABL1 P00519 1/20 0.44
LCK P06239 1/20 0.44
FGFR4 P22455 1/20 0.43
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
TTBK1 Q5TCY1 1/20 0.40
BRAF P15056 1/20 0.40
CHEK2 O96017 1/20 0.40
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417418 0.86 EGFR (0.61) EGFRFGFR4SCN5ASCN9APIK3CD
SCHEMBL27468871 0.78 CYP1A2 (0.52) MAP4K4CYP1A2CYP2C9CYP2C19ABL1
SCHEMBL4412993 0.78 EGFR (0.55) EGFRMAP4K4ABL1FGFR4SCN5A
SCHEMBL4147243 0.77 EGFR (0.60) EGFRFGFR4PIK3CDPIK3CA
SCHEMBL4412557 0.77 EGFR (0.61) EGFRABL1FGFR4PIK3CDPIK3CA
SCHEMBL5074400 0.77 EGFR (0.56) EGFRABL1FGFR4PIK3CDPIK3CA
SCHEMBL28292983 0.73 CYP2D6 (0.47) EGFRMAP4K4CYP1A2CYP2C9CYP2C19
SCHEMBL27399910 0.73 EGFR (0.65) EGFRFGFR4PIK3CDPIK3CA
SCHEMBL10715309 0.73 MAPT (0.54) CYP1A2CYP2C9CYP2C19SCN5ASCN9A
SCHEMBL29924283 0.73 RHEB (0.52) CYP1A2CYP2C9CYP2C19SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE41065-E1 Alkynl and azido-substituted 4-anilinoquinazolines PFIZER, INC. (US) 2009-12-29 US disclosed