SCHEMBL4412993

SCHEMBL4412993

Clc1ccccc1Oc1ccc2ncncc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.55
ABL1 P00519 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46
MAP4K4 O95819 1/20 0.45
FGFR4 P22455 1/20 0.45
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
KCNH2 Q12809 2/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
AR P10275 1/20 0.39
TDO2 P48775 1/20 0.39
TTBK1 Q5TCY1 1/20 0.38
TTBK2 Q6IQ55 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
MAPK14 Q16539 1/20 0.37
NOTUM Q6P988 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417418 0.79 EGFR (0.61) EGFRHTTFGFR4PIK3CDPIK3CA
SCHEMBL4412970 0.78 EGFR (0.56) EGFRABL1MAP4K4FGFR4PIK3CD
SCHEMBL24125011 0.74 NOTUM (0.46) EGFRALDH1A1KCNH2SCN5ASCN9A
SCHEMBL4412557 0.73 EGFR (0.61) EGFRABL1FGFR4PIK3CDPIK3CA
SCHEMBL5074400 0.72 EGFR (0.56) EGFRABL1FGFR4PIK3CDPIK3CA
SCHEMBL27399910 0.72 EGFR (0.65) EGFRFGFR4PIK3CDPIK3CAAR
SCHEMBL3372138 0.72 EGFR (1.00) EGFRALDH1A1FGFR4PIK3CDPIK3CA
SCHEMBL4418182 0.70 EGFR (0.47) EGFRALDH1A1HTTMAP4K4FGFR4
Hydrochloric Acid SCHEMBL28032872 0.70 EGFR (0.96) EGFRALDH1A1FGFR4PIK3CDPIK3CA
SCHEMBL7176453 0.70 DPP4 (0.53) ALDH1A1HTTKCNH2SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE41065-E1 Alkynl and azido-substituted 4-anilinoquinazolines PFIZER, INC. (US) 2009-12-29 US disclosed