SCHEMBL4413824

SCHEMBL4413824

Cn1cnc2c(=O)n(-c3ccc(F)cc3)c(C3CC(C(F)(F)F)C3)nc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.35
DRD1 P21728 5/20 0.34
DRD5 P21918 5/20 0.34
HKDC1 Q2TB90 2/20 0.34
KCNN3 Q9UGI6 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
TRPA1 O75762 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3178194 0.92 DRD1 (0.38) MAPK14DRD1DRD5ADORA3ADORA2A
SCHEMBL3178189 0.92 DRD1 (0.38) MAPK14DRD1DRD5ADORA3ADORA2A
SCHEMBL4506393 0.83 PIK3CD (0.38) MAPK14DRD1DRD5HKDC1SMN1; SMN2
SCHEMBL3179574 0.82 DRD1 (0.44) DRD1DRD5SMN1; SMN2PIK3CDPIK3CA
SCHEMBL3179577 0.82 DRD1 (0.44) DRD1DRD5SMN1; SMN2PIK3CDPIK3CA
SCHEMBL4791118 0.80 TRPV4 (0.35) PIK3CDPIK3CAPIK3CGPDE4APDE4B
SCHEMBL3169024 0.80 CTSS (0.36) DRD1DRD5
SCHEMBL3169031 0.80 CTSS (0.36) DRD1DRD5
SCHEMBL3177134 0.79 CDK1 (0.38) DRD1DRD5SMN1; SMN2TSHRPDE4A
SCHEMBL3177139 0.79 CDK1 (0.38) DRD1DRD5SMN1; SMN2TSHRPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO disclosed