SCHEMBL4415069

SCHEMBL4415069

Cc1ccc(NC(=O)c2cc(C#N)cc(N3CCCCC3)c2)cc1-c1cc(C(=O)NCc2ccccn2)on1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.47
SMO Q99835 2/20 0.47
TDP1 Q9NUW8 1/20 0.40
NPC1 O15118 1/20 0.39
RAF1 P04049 7/20 0.38
BRAF P15056 6/20 0.38
KDM4E B2RXH2 1/20 0.38
HSPB1 P04792 1/20 0.38
LYN P07948 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4408497 0.99 MAPK14 (0.48) MAPK14SMOTDP1NPC1RAF1
SCHEMBL4407770 0.94 MAPK14 (0.51) MAPK14SMORAF1BRAF
SCHEMBL4414281 0.89 MAPK14 (0.58) MAPK14SMONPC1RAF1BRAF
SCHEMBL4416214 0.88 MAPK14 (0.43) MAPK14NPC1RAF1BRAF
SCHEMBL4408184 0.87 MAPK14 (0.56) MAPK14SMORAF1BRAFLYN
SCHEMBL4418552 0.87 MAPK14 (0.44) MAPK14NPC1RAF1BRAF
SCHEMBL4409531 0.86 RAF1 (0.42) RAF1BRAF
SCHEMBL5604132 0.85 TEK (0.45) MAPK14NPC1RAF1BRAFKDM4E
SCHEMBL4409551 0.85 RAF1 (0.43) RAF1BRAF
SCHEMBL5593352 0.84 RAF1 (0.41) MAPK14NPC1RAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035005-A2 THERAPY USING CYTOKINE INHIBITORS Kemia, INC. (US) 2009-03-18 EP disclosed
WO-2007146712-A2 THERAPY USING CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-12-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed