SCHEMBL4415686

SCHEMBL4415686

CC(C)(C)OC(=O)N1CC2C[C@H]1CN2c1nc2c(C(=O)O)cccc2o1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
GPR119 Q8TDV5 1/20 0.43
HSD11B1 P28845 1/20 0.42
HDAC1 Q13547 1/20 0.42
HTR3A P46098 12/20 0.40
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
TGM1 P22735 1/20 0.37
MAPK8 P45983 1/20 0.37
SPR P35270 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1003663 0.91 PARP1 (0.46) PARP1GPR119HSD11B1HDAC1HTR3A
SCHEMBL1005642 0.79 HTR3A (0.45) PARP1GPR119HTR3A
SCHEMBL1005641 0.79 HTR3A (0.45) PARP1GPR119HTR3A
SCHEMBL1003480 0.79 ABCB1 (0.44) PARP1GPR119HTR3A
SCHEMBL1004366 0.79 ABCB1 (0.44) PARP1GPR119HTR3A
SCHEMBL1005752 0.78 NAAA (0.49) GPR119HDAC1HTR3AKCNH2
SCHEMBL1006345 0.77 NR1H3 (0.53) HTR3AKCNH2
SCHEMBL1006343 0.77 NR1H3 (0.53) HTR3AKCNH2
SCHEMBL1005424 0.77 HTR3A (0.47) PARP1GPR119HTR3AKCNH2
SCHEMBL1003499 0.77 HTR3A (0.47) PARP1GPR119HTR3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed