SCHEMBL4417850

SCHEMBL4417850

O=C1CC(CO)N(C(=O)c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.51
AVPR1A P37288 1/20 0.51
HPGD P15428 2/20 0.44
MAPK1 P28482 1/20 0.44
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
POLB P06746 2/20 0.41
SLC6A7 Q99884 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
RAB9A P51151 1/20 0.40
TSHR P16473 2/20 0.40
FASN P49327 1/20 0.40
ABCB1 P08183 1/20 0.40
SPHK2 Q9NRA0 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL301777 1.00 OXTR (0.51) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4414514 0.89 HPGD (0.42) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4414519 0.89 HPGD (0.42) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4419397 0.89 HPGD (0.44) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL8320159 0.89 HPGD (0.44) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4418365 0.88 HPGD (0.43) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4418361 0.88 HPGD (0.43) OXTRAVPR1AHPGDMAPK1HCRTR1
SCHEMBL4428848 0.86 AVPR1A (0.69) OXTRAVPR1AHCRTR1HCRTR2SLC6A7
SCHEMBL4428850 0.86 AVPR1A (0.69) OXTRAVPR1AHCRTR1HCRTR2SLC6A7
SCHEMBL13789901 0.85 SMN1; SMN2 (0.43) OXTRAVPR1AHPGDMAPK1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532109-B1 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS MERCK SERONO SA (CH) 2009-09-09 EP claimed
EP-1725526-B1 METHOD FOR PREPARING PYRROLIDINE OXIMES SERONO LAB (CH) 2007-12-12 EP claimed