SCHEMBL4419629

SCHEMBL4419629

CCC(=O)N(c1cccc(C(F)(F)F)c1)c1cnc(Oc2ccnc3cc(OC)c(OC)cc23)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.46
EGFR P00533 3/20 0.45
CSF1R P07333 3/20 0.45
MET P08581 3/20 0.44
MAPK14 Q16539 2/20 0.44
AURKA O14965 1/20 0.44
PIK3CA P42336 1/20 0.44
TEK Q02763 1/20 0.44
AURKB Q96GD4 1/20 0.44
AXL P30530 1/20 0.44
FGFR4 P22455 1/20 0.44
PDGFRA P16234 2/20 0.43
RET P07949 1/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
DDR1 Q08345 1/20 0.43
BRAF P15056 3/20 0.43
TNNI3K Q59H18 1/20 0.42
RAF1 P04049 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2203252 0.80 KDR (0.48) KDRMETAURKATEKAURKB
SCHEMBL378510 0.77 KDR (0.59) KDREGFRCSF1RMETMAPK14
SCHEMBL29693652 0.77 KDR (0.59) KDREGFRCSF1RMETMAPK14
SCHEMBL20525857 0.77 KDR (0.50) KDREGFRMETAURKATEK
SCHEMBL2364278 0.77 KDR (0.52) KDRCSF1RMETAURKATEK
SCHEMBL8554907 0.77 KDR (0.55) KDREGFRCSF1RMETMAPK14
SCHEMBL31324666 0.76 PDGFRB (0.62) KDRCSF1RMETMAPK14AURKA
SCHEMBL29693548 0.76 PDGFRB (0.62) KDRCSF1RMETMAPK14AURKA
SCHEMBL372681 0.76 PDGFRB (0.62) KDRCSF1RMETMAPK14AURKA
SCHEMBL20525836 0.76 AXL (0.49) KDREGFRMETAURKATEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170896-A1 c-Met modulators and methods of use EXELIXIS, INC. (US) 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170896-A1 c-Met modulators and methods of use FLT4, MET, FLT1 KDR 5/4885EGFR 166/4885CSF1R 214/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.