SCHEMBL4420558

SCHEMBL4420558

O=C(O)N1CCC2(CCn3c(nc(-c4ccncn4)cc3=O)N2)C1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.39
CYP46A1 Q9Y6A2 2/20 0.35
CYP2D6 P10635 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4420553 1.00 GSK3B (0.39) GSK3BCYP46A1CYP2D6
SCHEMBL5559168 0.87 GSK3B (0.40) GSK3B
SCHEMBL5559165 0.87 GSK3B (0.40) GSK3B
SCHEMBL4429026 0.87 ALDH1A1 (0.38) GSK3BCYP46A1
SCHEMBL4420810 0.85 CYP2C9 (0.46) GSK3BCYP2D6
SCHEMBL4421898 0.82 GSK3B (0.53) GSK3BCYP2D6
SCHEMBL4416863 0.81 GSK3B (0.42) GSK3B
SCHEMBL4418095 0.80 ALDH1A1 (0.39) GSK3BCYP46A1
SCHEMBL3560210 0.79 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL4428471 0.74 CDC7 (0.44) GSK3BCYP46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547705-B2 Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives SANOFI-AVENTIS (FR) 2009-06-16 US disclosed