SCHEMBL4429026

SCHEMBL4429026

O=C(O)N1CCC2(CCn3c(nc(-c4ccncc4)cc3=O)N2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
CYP2C9 P11712 1/20 0.35
USP19 O94966 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35
GSK3B P49841 9/20 0.34
CDC7 O00311 4/20 0.34
PIM1 P11309 3/20 0.34
HIPK2 Q9H2X6 3/20 0.34
CLK4 Q9HAZ1 3/20 0.34
ROCK2 O75116 2/20 0.34
MAP4K4 O95819 2/20 0.34
PRKACA P17612 2/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4418095 0.94 ALDH1A1 (0.39) ALDH1A1TSHRKDM4EGLAHTT
SCHEMBL4420553 0.87 GSK3B (0.39) GSK3BCYP46A1
SCHEMBL4420558 0.87 GSK3B (0.39) GSK3BCYP46A1
SCHEMBL4428471 0.86 CDC7 (0.44) ALDH1A1TSHRKDM4EGLAHTT
SCHEMBL4421551 0.82 CDC7 (0.46) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL4418556 0.81 GSK3B (0.42) KDM5BGSK3BCDC7PIM1HIPK2
SCHEMBL4867552 0.77 KDM5B (0.41) KDM5BGSK3BCDC7PIM1HIPK2
SCHEMBL5559165 0.74 GSK3B (0.40) ALDH1A1KDM4EGSK3B
SCHEMBL4420810 0.72 CYP2C9 (0.46) ALDH1A1TSHRSMN1; SMN2CYP2C9GSK3B
SCHEMBL4865645 0.72 KDM5B (0.46) KDM5BGSK3BCDC7PIM1HIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547705-B2 Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives SANOFI-AVENTIS (FR) 2009-06-16 US disclosed