SCHEMBL4423456

SCHEMBL4423456

CCOc1cc(C(=O)[C@@H]2C(=O)c3cc(-c4ccnc(C(=O)O)c4)ccc3OC23CCNCC3)cc(OCC)c1-c1cnn(C)c1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.34
GSK3B P49841 6/20 0.33
DYRK1A Q13627 6/20 0.33
WNT1 P04628 5/20 0.33
ADH5 P11766 3/20 0.33
SSTR5 P35346 3/20 0.32
CSF1R P07333 1/20 0.32
TTK P33981 2/20 0.32
MAP4K4 O95819 1/20 0.31
MAPK8 P45983 1/20 0.31
IRAK4 Q9NWZ3 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4416789 0.90 ACACB (0.38) GSK3BDYRK1AWNT1ADH5SSTR5
SCHEMBL4427891 0.88 SSTR5 (0.37) ADH5SSTR5CSF1RMAP4K4IRAK4
SCHEMBL4424719 0.88 CYP2D6 (0.32) GSK3BDYRK1AWNT1SSTR5IRAK4
SCHEMBL4412902 0.88 ACACB (0.41) GSK3BDYRK1AWNT1ADH5SSTR5
SCHEMBL2599528 0.87 SSTR5 (0.39) GSK3BDYRK1AWNT1SSTR5
SCHEMBL4412864 0.87 SSTR5 (0.34) GSK3BDYRK1AWNT1ADH5SSTR5
SCHEMBL4423563 0.86 TTK (0.33) GSK3BDYRK1AWNT1ADH5TTK
SCHEMBL4427980 0.86 GSK3B (0.33) GSK3BDYRK1AWNT1SSTR5CSF1R
SCHEMBL4418731 0.85 GSK3B (0.32) GSK3BDYRK1AWNT1SSTR5IRAK4
SCHEMBL4423082 0.84 IRAK4 (0.33) GSK3BDYRK1AWNT1CSF1RTTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP claimed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO claimed
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed