SCHEMBL4423528

SCHEMBL4423528

FC(F)(F)c1ccc2c(c1)Sc1ccccc1[N]2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYBB P04839 1/20 0.51
NOX3 Q9HBY0 1/20 0.51
NOX4 Q9NPH5 1/20 0.51
NOX1 Q9Y5S8 1/20 0.51
PTPN5 P54829 1/20 0.40
TRPA1 O75762 1/20 0.39
TP53 P04637 3/20 0.39
TSHR P16473 3/20 0.39
NPC1 O15118 2/20 0.39
CYP1A2 P05177 2/20 0.39
ABCB1 P08183 2/20 0.39
HTR1A P08908 2/20 0.39
ADRA2A P08913 2/20 0.39
ADORA3 P0DMS8 2/20 0.39
CYP2D6 P10635 2/20 0.39
CHRM1 P11229 2/20 0.39
DRD1 P21728 2/20 0.39
SLC6A2 P23975 2/20 0.39
MAPK1 P28482 2/20 0.39
SLC6A4 P31645 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2748095 0.93 CYBB (0.57) CYBBNOX3NOX4NOX1PTPN5
SCHEMBL24828 0.79 TRPA1 (0.54) NOX1TRPA1NPC1CYP1A2HTR1A
SCHEMBL28924686 0.78 CYBB (0.65) CYBBNOX3NOX4NOX1PTPN5
SCHEMBL28367426 0.76 GPR3 (0.44) TSHRCHRM1MAPK1MAPTALDH1A1
SCHEMBL28372461 0.72 GPR3 (0.49) CYBBNOX3NOX4NOX1TSHR
SCHEMBL9507729 0.71 PTPN5 (0.58) CYBBNOX3NOX4NOX1PTPN5
SCHEMBL9511171 0.71 PTPN5 (0.58) CYBBNOX3NOX4NOX1PTPN5
SCHEMBL10372692 0.69 NOX1 (0.84) CYBBNOX3NOX4NOX1NPC1
SCHEMBL11753992 0.69 CYBB (0.54) CYBBNOX3NOX4NOX1PTPN5
SCHEMBL30811565 0.69 NOX1 (0.84) CYBBNOX3NOX4NOX1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625951-B2 Stimuli-responsive hydrogel microdomes integrated with genetically engineered proteins for high-throughput screening of pharmaceuticals UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2009-12-01 US disclosed
US-20050208469-A1 Stimuli-responsive hydrogel microdomes integrated with genetically engineered proteins for high-throughput screening of pharmaceuticals UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION 2005-09-22 US disclosed