SCHEMBL4425287

SCHEMBL4425287

CP(C)(=O)CCOC(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
CHRM2 P08172 2/20 0.46
CHRM4 P08173 2/20 0.46
CHRM5 P08912 2/20 0.46
CHRM1 P11229 2/20 0.46
CHRM3 P20309 2/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 2/20 0.46
TSHR P16473 2/20 0.46
HTR1A P08908 1/20 0.46
CYP2C19 P33261 1/20 0.46
CHRNA7 P36544 1/20 0.46
ALOX15 P16050 1/20 0.44
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CA4 P22748 3/20 0.33
HSD17B10 Q99714 1/20 0.33
CA1 P00915 2/20 0.32
CA5A P35218 2/20 0.32
CA5B Q9Y2D0 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11763356 0.86 LMNA (0.43) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL10308490 0.78 ALDH1A1 (0.46) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL1976413 0.78 LMNA (0.43) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL2547540 0.73 LMNA (0.57) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL499368 0.72
SCHEMBL9846963 0.71 TSHR (0.54) TSHRHSD17B10
SCHEMBL14895398 0.70
Ammonia Solution, Strong SCHEMBL27654016 0.70
SCHEMBL30525718 0.70 LMNA (0.62) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL41800 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049124-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP disclosed
WO-2008010985-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2008-01-24 WO disclosed