SCHEMBL4426472

SCHEMBL4426472

O=C1COC(c2ccccc2)=NN1Cc1cc[c]cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
THRB P10828 1/20 0.43
MAOB P27338 2/20 0.40
LMNA P02545 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
PGR P06401 1/20 0.40
CYP2D6 P10635 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1080923 0.82 GAA (0.45) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL1078929 0.79 KMT2A (0.35) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL1078878 0.77 KMT2A (0.44) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL1177873 0.76 KMT2A (0.39) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL3695678 0.75 KMT2A (0.43) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL7601875 0.75 KMT2A (0.38) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL1070118 0.75 KMT2A (0.38) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL517151 0.73 KMT2A (0.37) KMT2AALDH1A1GAATHRBMAOB
SCHEMBL517093 0.73 ALOX5 (0.39) KMT2AMAOBCYP2D6
SCHEMBL1079340 0.73 MAOB (0.37) KMT2AMAOBLMNAPGRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127338-A1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-10-22 WO disclosed