SCHEMBL4426737

SCHEMBL4426737

Brc1ccc(Nc2ccnc(Nc3ccc(Br)cc3)n2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 8/20 0.69
NPC1 O15118 3/20 0.69
MAPT P10636 3/20 0.69
MAPK1 P28482 3/20 0.69
RAB9A P51151 3/20 0.69
MEN1 O00255 2/20 0.69
LMNA P02545 2/20 0.69
KMT2A Q03164 2/20 0.69
ALOX12 P18054 1/20 0.69
CHEK1 O14757 1/20 0.68
IKBKB O14920 1/20 0.68
PDPK1 O15530 1/20 0.68
CHEK2 O96017 1/20 0.68
PRKCG P05129 1/20 0.68
CDK1 P06493 1/20 0.68
LYN P07948 1/20 0.68
KIT P10721 1/20 0.68
PIM1 P11309 1/20 0.68
FGFR1 P11362 1/20 0.68
FGFR3 P22607 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1321961 0.81 AURKA (1.00) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL379222 0.81 AURKA (0.69) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL440486 0.81 AURKA (1.00) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL31337079 0.80 ROCK1 (0.69) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL5263722 0.80 PIK3CA (0.48) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL1120994 0.78 PIK3CG (0.51) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL23887662 0.77 KDR (0.47) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL30086805 0.77 KDR (0.47) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL5384269 0.76 AURKA (0.87) AURKANPC1MAPTMAPK1RAB9A
SCHEMBL4621303 0.76 NPC1 (0.87) AURKANPC1MAPTMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648524-B1 USE OF SUBSTITUTED 2,4-BIS (ALKYLAMINO) PYRIMIDINES OR -QUINAZOLINES AS ANTIMICROBIALS CIBA HOLDING INC (CH) 2009-01-14 EP disclosed