SCHEMBL4428229

SCHEMBL4428229

COC(=O)c1cc(C(c2ccccc2)c2ccccc2)n(C)c(=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
PPARA Q07869 3/20 0.46
GAA P10253 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PPARG P37231 2/20 0.41
KDM4E B2RXH2 1/20 0.41
OPRD1 P41143 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
CASP3 P42574 2/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16345385 0.73 FGFR1 (0.55) TSHRGAAALDH1A1KDM4ESMN1; SMN2
SCHEMBL2896391 0.72 CYP1A2 (0.50) TSHRGAAL3MBTL1ALDH1A1KDM4E
SCHEMBL10796231 0.72 CA12 (0.52) TSHRGAAL3MBTL1ALDH1A1KDM4E
SCHEMBL4986643 0.71 OPRD1 (0.47) TSHRPPARAGAAL3MBTL1ALDH1A1
SCHEMBL4433925 0.71 TSHR (0.46) TSHRPPARAGAAL3MBTL1ALDH1A1
SCHEMBL14972272 0.70 MAPK1 (0.50) TSHRPPARAGAAL3MBTL1ALDH1A1
SCHEMBL14967035 0.70 MAPK1 (0.50) TSHRPPARAGAAL3MBTL1ALDH1A1
SCHEMBL22579467 0.70 CA12 (0.46) TSHRGAAL3MBTL1ALDH1A1KDM4E
SCHEMBL27878777 0.67 TSHR (0.68) TSHRGAAL3MBTL1ALDH1A1KDM4E
SCHEMBL22556827 0.67 AR (0.43) TSHRGAAL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed