SCHEMBL4428254

SCHEMBL4428254

O=C(O)c1ccc(C(c2ccc(C(F)(F)F)cc2)c2ccc(C(F)(F)F)cc2)[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 8/20 0.49
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 2/20 0.42
UCHL1 P09936 1/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
SRD5A2 P31213 1/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX12 P18054 1/20 0.38
KMT2A Q03164 1/20 0.38
USP2 O75604 1/20 0.38
CYP2C19 P33261 1/20 0.38
ACP3 P15309 1/20 0.37
CYP2C8 P10632 1/20 0.37
SORT1 Q99523 1/20 0.36
PDE2A O00408 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438805 0.84 HSD17B2 (0.48) HSD17B2KDM4EPDE2A
SCHEMBL4427252 0.82 KDM4E (0.53) HSD17B2KDM4EALDH1A1MEN1KMT2A
SCHEMBL14931973 0.75 KDM4E (0.66) HSD17B2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4429520 0.74 KDM4E (0.42) HSD17B2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4439660 0.73 KDM4E (0.41) KDM4ECES2CES1MEN1KMT2A
SCHEMBL3071414 0.73 KDM4E (0.49) HSD17B2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4379536 0.71 KDM5A (0.54) HSD17B2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4430946 0.70 HSD17B2 (0.46) HSD17B2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL5124119 0.70 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL3077344 0.70 HSD17B2 (0.52) HSD17B2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed