SCHEMBL4429182

SCHEMBL4429182

COC(=O)/C=C/c1ccc(C(=O)OC(=O)c2ccc(C=O)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.62
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
TYR P14679 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA14 Q9ULX7 1/20 0.58
MAPT P10636 5/20 0.55
KDM4E B2RXH2 3/20 0.55
PTPN1 P18031 2/20 0.51
APP P05067 2/20 0.50
TTR P02766 1/20 0.50
LMNA P02545 3/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 2/20 0.49
EPHX2 P34913 1/20 0.47
ESR1 P03372 1/20 0.46
MEN1 O00255 1/20 0.46
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20653 0.88 CA12 (0.72) ALDH1A1CA12CA1CA2TYR
SCHEMBL20654 0.88 CA12 (0.72) ALDH1A1CA12CA1CA2TYR
Hydrochloric Acid SCHEMBL724882 0.87 CA12 (0.70) ALDH1A1CA12CA1CA2TYR
Hydrochloric Acid SCHEMBL724881 0.87 CA12 (0.70) ALDH1A1CA12CA1CA2TYR
SCHEMBL4429187 0.86 ALDH1A1 (0.61) ALDH1A1CA12CA1CA2TYR
SCHEMBL4429179 0.86 ALDH1A1 (0.61) ALDH1A1CA12CA1CA2TYR
SCHEMBL1133144 0.85 CA12 (0.68) ALDH1A1CA12CA1CA2TYR
SCHEMBL11332365 0.85 CA12 (0.68) ALDH1A1CA12CA1CA2TYR
SCHEMBL71224 0.81 CA12 (0.84) ALDH1A1CA12CA1CA2TYR
SCHEMBL475274 0.81 ALDH1A1 (0.69) ALDH1A1MAPTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069291-A1 HDAC INHIBITORS Chroma Therapeutics Limited (GB) 2009-06-17 EP disclosed
WO-2008040934-A1 HDAC INHIBITORS CHROMA THERAPEUTICS LTD. (GB) 2008-04-10 WO disclosed