SCHEMBL4430700

SCHEMBL4430700

O=C(O)C1CCC2(CC=NC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.35
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
GRM2 Q14416 2/20 0.35
GRM3 Q14832 2/20 0.35
GRM4 Q14833 2/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 2/20 0.35
CYP1A2 P05177 1/20 0.35
ALOX15 P16050 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GRM8 O00222 1/20 0.35
GRM6 O15303 1/20 0.35
GRM5 P41594 1/20 0.35
MTOR P42345 1/20 0.35
GRM1 Q13255 1/20 0.35
PLCB1 Q9NQ66 1/20 0.35
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441504 0.84 CYP3A4 (0.31)
SCHEMBL4436006 0.81 CYP2C19 (0.54) CYP2C19CYP1A2ALOX15GABRPGABRD
SCHEMBL8004566 0.75 CYP2C19 (0.52) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL848416 0.73 CYP2C19 (0.50) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL8810863 0.69 CYP2C19 (0.46) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL4532840 0.69 CYP2C19 (0.46) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL515587 0.67 CYP2C19 (0.44) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL11646566 0.66 CYP2C19 (0.62) CYP2C19ITGB3ITGA2BGRM2GRM3
SCHEMBL23603993 0.66 CYP2C19 (0.42) CYP2C19ITGB3ITGA2BGRM2GRM3
Hydrochloric Acid SCHEMBL11636408 0.66 CYP2C19 (0.42) CYP2C19ITGB3ITGA2BGRM2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124944-A1 PYRAZOLO (3, 4-B) PYRIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2009-12-02 EP claimed
WO-2008111010-A1 PYRAZOLO (3, 4-B) PYRIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2008-09-18 WO claimed