SCHEMBL4431360

SCHEMBL4431360

CNC(=O)C(NCCC(c1ccc(C(F)(F)F)nc1)c1cc(Cl)ccc1OC)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 12/20 0.42
IGF1R P08069 1/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CTSA P10619 2/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4440486 1.00 P2RX7 (0.42) P2RX7IGF1RMAPK1ALDH1A1CTSA
SCHEMBL4440271 0.93 P2RX7 (0.40) P2RX7MAPK1CTSAEPHX2
SCHEMBL4441753 0.88 P2RX7 (0.40) P2RX7MAPK1EPHX2
SCHEMBL4428035 0.87 P2RX7 (0.45) P2RX7MAPK1EPHX2
SCHEMBL4429693 0.87 P2RX7 (0.45) P2RX7MAPK1EPHX2
SCHEMBL4441204 0.86 P2RX7 (0.41) P2RX7MAPK1EPHX2
SCHEMBL4434611 0.86 P2RX7 (0.41) P2RX7MAPK1EPHX2
SCHEMBL4441632 0.86 P2RX7 (0.41) P2RX7MAPK1EPHX2
SCHEMBL4432133 0.86 P2RX7 (0.41) P2RX7ALDH1A1
SCHEMBL4432125 0.86 P2RX7 (0.41) P2RX7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed