SCHEMBL4432174

SCHEMBL4432174

CNC(=O)[C@@H](NCC[C@H](c1ccc(C(F)(F)F)cc1)c1ccc(F)c(OC(F)(F)F)c1)c1ccc(C)cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CCR2 P41597 4/20 0.35
CASR P41180 1/20 0.35
TACR1 P25103 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
UTS2R Q9UKP6 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
ALOX5 P09917 3/20 0.34
EPHX2 P34913 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441647 0.94 KDM4E (0.42) KDM4ECCR2CASRTACR1ALDH1A1
SCHEMBL4428140 0.90 CTSA (0.37) CTSACNR1CNR2CASRUTS2R
SCHEMBL4431321 0.90 CTSA (0.37) CTSACNR1CNR2CASRUTS2R
SCHEMBL4427927 0.84 CNR1 (0.51) KDM4ECNR1CNR2CCR2CASR
SCHEMBL4434552 0.84 CNR1 (0.51) KDM4ECNR1CNR2CCR2CASR
SCHEMBL4441795 0.82 KDM4E (0.46) KDM4ECNR1CNR2CCR2TACR1
SCHEMBL4430647 0.82 KDM4E (0.46) KDM4ECNR1CNR2CCR2TACR1
SCHEMBL4431479 0.82 ALOX5 (0.39) CNR2CCR2CASRTACR1ALOX5
SCHEMBL4432382 0.82 ALOX5 (0.39) CNR2CCR2CASRTACR1ALOX5
SCHEMBL4441777 0.81 KDM4E (0.46) KDM4ECCR2TACR1ALDH1A1CTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed