SCHEMBL4432347

SCHEMBL4432347

COc1ccc(C(C(C)=O)c2ccc(C)cc2)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
MAPT P10636 2/20 0.50
LMNA P02545 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HTT P42858 1/20 0.49
CTNNB1 P35222 1/20 0.49
WNT3A P56704 1/20 0.49
ACHE P22303 2/20 0.48
POLB P06746 1/20 0.46
PPARG P37231 1/20 0.44
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44
EPHX2 P34913 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16973606 0.87 TDP1 (0.51) ALDH1A1MAPTLMNAACHEPOLB
SCHEMBL4434628 0.82 AKR1C3 (0.51) MAPTACHEPPARGPPARDPPARA
SCHEMBL8295353 0.80 NR1H4 (0.45) ALDH1A1LMNAKDM4EACHEPPARG
SCHEMBL8145960 0.78 ACHE (0.46) ALDH1A1MAPTLMNAKDM4EACHE
SCHEMBL16246442 0.77 TUBB4A (0.46) ALDH1A1KDM4EHTTACHEPPARG
Acetone SCHEMBL8119850 0.77 STAT3 (0.42) ALDH1A1LMNAHTTACHEPOLB
SCHEMBL15540879 0.76 TSHR (0.56) HTTACHECYP3A4TSHRKMT2A
SCHEMBL16867628 0.76 ACHE (0.53) ACHEPPARGPPARDPPARACYP1A2
SCHEMBL16867623 0.76 ACHE (0.53) ACHEPPARGPPARDPPARACYP1A2
SCHEMBL19365873 0.76 ACHE (0.53) ACHEPPARGPPARDPPARACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed