SCHEMBL4432890

SCHEMBL4432890

COc1cccc(NCCCc2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.49
MTNR1B P49286 3/20 0.49
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KMT2A Q03164 3/20 0.47
TDP1 Q9NUW8 1/20 0.47
MCHR1 Q99705 1/20 0.47
GAK O14976 1/20 0.46
MEN1 O00255 2/20 0.45
ACP1 P24666 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HTT P42858 1/20 0.44
CASR P41180 2/20 0.44
ADRB2 P07550 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581197 0.93 TDP1 (0.51) MTNR1AMTNR1BHDAC1HDAC8HDAC6
SCHEMBL4433139 0.85 MAPT (0.57) KMT2AMCHR1MEN1ACP1GAA
Hydrochloric Acid SCHEMBL4441377 0.83 MAPT (0.56) KMT2AMCHR1MEN1ACP1GAA
SCHEMBL1582274 0.83 ACP1 (0.51) MTNR1AMTNR1BHDAC1HDAC8HDAC6
SCHEMBL11117603 0.83 MAPT (0.56) MTNR1AMTNR1BKMT2ATDP1GAK
SCHEMBL4434676 0.81 MCHR1 (0.49) KMT2ATDP1MCHR1MEN1KDM4E
SCHEMBL15130900 0.80 CASR (0.63) KMT2AMEN1HTTCASR
SCHEMBL3648940 0.80 ALDH1A1 (0.44) ACP1HTTGAAMAPTSIRT2
SCHEMBL27610543 0.79 ALDH1A1 (0.53) HDAC1HDAC8MCHR1MAPT
SCHEMBL11114174 0.79 MTNR1A (0.66) MTNR1AMTNR1BKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed