SCHEMBL4433135

SCHEMBL4433135

COC(=O)c1ccc([N+](=O)[O-])c(C(C(=O)O)C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.53
ALDH1A1 P00352 3/20 0.48
AR P10275 1/20 0.46
PELP1 Q8IZL8 1/20 0.46
KMT2A Q03164 2/20 0.46
HPGD P15428 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PKM P14618 1/20 0.45
AKR1C4 P17516 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
AKR1C1 Q04828 1/20 0.45
LMNA P02545 1/20 0.44
ERN1 O75460 1/20 0.44
TSHR P16473 1/20 0.44
POLB P06746 2/20 0.44
CASP6 P55212 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4446049 1.00 VCAM1 (0.53) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL8768519 0.84 VCAM1 (0.46) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL4125942 0.84 VCAM1 (0.55) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL29625012 0.84 VCAM1 (0.55) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL7087722 0.84 VCAM1 (0.55) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL5004220 0.83 VCAM1 (0.51) VCAM1ALDH1A1ARPELP1KMT2A
SCHEMBL5734347 0.80 VCAM1 (0.68) VCAM1ALDH1A1KMT2AHPGDNPSR1
SCHEMBL9652429 0.79 AKR1C3 (0.49) ALDH1A1KMT2AHPGDAKR1C4AKR1C3
SCHEMBL1291038 0.79 MAPK1 (0.59) VCAM1ALDH1A1KMT2AHPGDNPSR1
SCHEMBL29946151 0.79 MAPK1 (0.59) VCAM1ALDH1A1KMT2AHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121656-A1 INHIBITORS OF SERINE PALMITOYLTRANSFERASE Pfizer Products Inc. (US) 2009-11-25 EP disclosed
WO-2008084300-A1 INHIBITORS OF SERINE PALMITOYLTRANSFERASE PFIZER PRODUCTS INC. (US) 2008-07-17 WO disclosed
US-5872280-A RESPIRATORY SYSTEM DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1999-02-16 US disclosed