SCHEMBL4433402

SCHEMBL4433402

CCOC(=O)CNC(=O)C1CCCN1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
HSD17B10 Q99714 1/20 0.47
POLB P06746 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MMP2 P08253 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
FAP Q12884 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
FKBP1A P62942 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LTA4H P09960 1/20 0.40
NPC1 O15118 1/20 0.40
F2 P00734 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209842 1.00 TSHR (0.47) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL4436777 0.84 SMN1; SMN2 (0.60) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL18374165 0.84 SMN1; SMN2 (0.60) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL6354140 0.83 PREP (0.44) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL6357029 0.83 ALDH1A1 (0.52) TSHRKDM4EGAAHSD17B10MMP2
SCHEMBL6355254 0.82 GAA (0.46) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL29596119 0.81 TSHR (0.42) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL6355253 0.81 GAA (0.48) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL29735871 0.81 GAA (0.48) TSHRKDM4EGAAHSD17B10POLB
SCHEMBL5646661 0.81 RAB9A (0.41) KDM4EGAAHSD17B10POLBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed
EP-2121603-A2 6' SUBSTITUTED INDOLE AND INDAZOLE DERIVATIVES HAVING 5-HT6 RECEPTOR AFFINITY Memory Pharmaceuticals Corporation (US) 2009-11-25 EP disclosed
WO-2008101247-A2 6 ' SUBSTITUTED INDOLE AND INDAZOLE DERIVATIVES HAVING 5-HT6 RECEPTOR AFFINITY MEMORY PHARMACEUTICALS CORPORATION (US) 2008-08-21 WO disclosed