SCHEMBL4434465

SCHEMBL4434465

CON(C)C(=O)C1Cc2ccccc2N1C(=O)OCc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
OPRM1 P35372 3/20 0.43
OPRL1 P41146 3/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9964896 1.00 NPC1 (0.46) NPC1RAB9AL3MBTL1OPRM1OPRL1
SCHEMBL5764293 0.84 DRD2 (0.53) NPC1RAB9AL3MBTL1
SCHEMBL24582713 0.83 NPC1 (0.54) NPC1RAB9AL3MBTL1
SCHEMBL1000224 0.83 NPC1 (0.54) NPC1RAB9AL3MBTL1
SCHEMBL4442416 0.83 OPRM1 (0.47) OPRM1OPRL1
SCHEMBL3208272 0.83 NPC1 (0.54) NPC1RAB9AL3MBTL1
SCHEMBL1150621 0.82 NPC1 (0.46) NPC1RAB9AL3MBTL1PTGDR2TMEM97
SCHEMBL31092767 0.81 OPRL1 (0.41) OPRM1OPRL1
SCHEMBL31092768 0.81 OPRL1 (0.41) OPRM1OPRL1
SCHEMBL7036798 0.81 PTPN1 (0.52) NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134721-A1 ANTIMICROBIAL HETEROCYCLIC COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS Micurx Pharmaceuticals, Inc. (US) 2009-12-23 EP disclosed
WO-2008108988-A1 ANTIMICROBIAL HETEROCYCLIC COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (US) 2008-09-12 WO disclosed