SCHEMBL4434677

SCHEMBL4434677

COc1ccc(C(CCN)c2ccc(C(F)(F)F)cc2)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 4/20 0.45
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 2/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KCNK2 O95069 1/20 0.44
KCNH2 Q12809 1/20 0.44
CACNA1C Q13936 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
PPARD Q03181 2/20 0.41
PPARA Q07869 2/20 0.41
CYP19A1 P11511 1/20 0.40
RORC P51449 1/20 0.40
ACHE P22303 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433951 0.86 AKR1C3 (0.50) CASRAKR1C3AKR1C2MEN1KMT2A
SCHEMBL4433142 0.82 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL4441454 0.82 MEN1 (0.60) MEN1KMT2AMAPK1PPARDPPARA
Hydrochloric Acid SCHEMBL4441383 0.81 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL4430515 0.81 PDE4A (0.48) MEN1KMT2APPARDPPARAACHE
SCHEMBL4432755 0.81 AKR1C3 (0.51) AKR1C3AKR1C2PPARDPPARARORC
SCHEMBL4432893 0.81 SLC6A2 (0.51) CASRSLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL4441719 0.80 AKR1C3 (0.46) CASRAKR1C3AKR1C2MEN1KMT2A
SCHEMBL14387383 0.78 SLC6A2 (0.48) CASRSLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL4434646 0.78 AKR1C3 (0.45) CASRAKR1C3AKR1C2MAPK1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed