SCHEMBL4433142

SCHEMBL4433142

COc1ccc(C(CCN)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.55
SLC6A4 P31645 3/20 0.55
SLC6A3 Q01959 3/20 0.55
KCNH2 Q12809 3/20 0.55
KCNK2 O95069 2/20 0.55
CACNA1C Q13936 2/20 0.55
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
BACE1 P56817 2/20 0.50
ALDH1A1 P00352 1/20 0.49
SLC7A5 Q01650 4/20 0.48
CACNA1A O00555 1/20 0.46
CACNA2D1 P54289 1/20 0.46
CACNB1 Q02641 1/20 0.46
NPC1 O15118 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 2/20 0.45
MTOR P42345 2/20 0.45
RAB9A P51151 2/20 0.45
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4441383 0.98 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3KCNH2KCNK2
SCHEMBL5947827 0.87 KMT2A (0.65) MEN1KMT2AALDH1A1CYP2D6CYP2C19
SCHEMBL4432893 0.86 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3KCNH2KCNK2
SCHEMBL4441835 0.84 CACNA1A (0.48) SLC6A4MEN1KMT2ABACE1CACNA1A
SCHEMBL4434677 0.82 CASR (0.45) SLC6A2SLC6A4SLC6A3KCNH2KCNK2
SCHEMBL4432789 0.82 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3KCNH2KCNK2
SCHEMBL4435726 0.82 KMT2A (0.61) MEN1KMT2AALDH1A1CYP2D6CYP2C19
SCHEMBL5161949 0.82 HRH1 (0.67) SLC6A2SLC6A4SLC6A3KCNH2KCNK2
SCHEMBL10973267 0.82 HRH1 (0.67) SLC6A2SLC6A4MEN1KMT2AALDH1A1
SCHEMBL4440597 0.80 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3KCNH2KCNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed