SCHEMBL4434646

SCHEMBL4434646

COc1ccc(C(CCO)c2ccc(C(F)(F)F)cc2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.45
AKR1C2 P52895 3/20 0.45
CASR P41180 5/20 0.44
PDE2A O00408 3/20 0.40
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
KIF11 P52732 1/20 0.39
RORC P51449 1/20 0.39
CYP19A1 P11511 2/20 0.39
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433951 0.89 AKR1C3 (0.50) AKR1C3AKR1C2CASRMAPK1RORC
SCHEMBL4441835 0.80 CACNA1A (0.48) AKR1C3AKR1C2LMNAMAPK1HTT
SCHEMBL4434677 0.78 CASR (0.45) AKR1C3AKR1C2CASRMAPK1RORC
SCHEMBL3733088 0.77 TMEM97 (0.46) CASRPDE2A
SCHEMBL23960431 0.77 CYP19A1 (0.54) AKR1C3AKR1C2CYP19A1
SCHEMBL10667796 0.73 KIF11 (0.49) PDE2ALMNAMAPK1HTTRAB9A
SCHEMBL4441719 0.72 AKR1C3 (0.46) AKR1C3AKR1C2CASRMAPK1
SCHEMBL4432755 0.71 AKR1C3 (0.51) AKR1C3AKR1C2RORC
SCHEMBL13906295 0.70 CYP17A1 (0.56) CASRRAB9AKIF11
SCHEMBL15561617 0.69 LMNA (0.45) PDE2ALMNAMAPK1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed