SCHEMBL4434798

SCHEMBL4434798

CCc1ccccc1-c1cccc(C(N)=O)c1CC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
PARP1 P09874 3/20 0.42
FGFR1 P11362 1/20 0.41
FGFR2 P21802 1/20 0.41
FGFR4 P22455 1/20 0.41
FGFR3 P22607 1/20 0.41
SLC9A1 P19634 1/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLCN2 P51788 1/20 0.40
DPP4 P27487 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NR1I2 O75469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL528444 0.86 BCAT2 (0.55) BCAT2KEAP1NFE2L2PARP1FGFR1
SCHEMBL72113 0.86 PARP1 (0.49) BCAT2KEAP1NFE2L2PARP1MAPT
SCHEMBL4065283 0.85 MYC (0.47) BCAT2KEAP1NFE2L2PARP1FGFR1
Charcoal, Activated SCHEMBL9345241 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1MAPT
Hydrochloric Acid SCHEMBL7467552 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1MAPT
SCHEMBL6321332 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1MAPT
Fluoride SCHEMBL28693457 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1MAPT
Hydrochloric Acid SCHEMBL8527465 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1MAPT
SCHEMBL5524497 0.84 PARP1 (0.47) BCAT2KEAP1NFE2L2PARP1FGFR1
SCHEMBL4439618 0.83 BCAT2 (0.62) BCAT2KEAP1NFE2L2PARP1FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121621-A1 LXR AND FXR MODULATORS Exelixis, Inc. (US) 2009-11-25 EP disclosed
WO-2008073825-A1 LXR AND FXR MODULATORS EXELIXIS, INC. (US) 2008-06-19 WO disclosed