SCHEMBL4435099

SCHEMBL4435099

C/C=C(/C[C@H]1COC(C)(C)N1C(=O)OC(C)(C)C)c1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.50
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SPHK1 Q9NYA1 1/20 0.39
STS P08842 2/20 0.36
HSD11B2 P80365 1/20 0.35
ATM Q13315 1/20 0.34
GPR119 Q8TDV5 2/20 0.34
DRD2 P14416 1/20 0.34
GABRA5 P31644 1/20 0.33
VEGFA P15692 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433026 0.89 KDM4E (0.43) BRD4MEN1KMT2ASPHK1STS
SCHEMBL3616035 0.80 BRD4 (0.49) BRD4MEN1KMT2AHTTSMN1; SMN2
SCHEMBL3616039 0.80 BRD4 (0.49) BRD4MEN1KMT2AHTTSMN1; SMN2
SCHEMBL3616041 0.80 BRD4 (0.49) BRD4MEN1KMT2AHTTSMN1; SMN2
SCHEMBL18959547 0.79 BRD4 (0.47) BRD4MEN1KMT2AHTTSMN1; SMN2
SCHEMBL1833586 0.78 BRD4 (0.47) BRD4MEN1KMT2ASPHK1GPR119
SCHEMBL1833587 0.78 BRD4 (0.47) BRD4MEN1KMT2ASPHK1GPR119
SCHEMBL3838091 0.77 BRD4 (0.47) BRD4MEN1KMT2ASTS
SCHEMBL3838083 0.77 BRD4 (0.47) BRD4MEN1KMT2ASTS
SCHEMBL6486940 0.77 BRD4 (0.46) BRD4MEN1KMT2AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114906-A1 NOVEL 2-AMINOOXAZOLINES AS TAAR1 LIGANDS FOR CNS DISORDERS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008092785-A1 NOVEL 2-AMINOOXAZOLINES AS TAAR1 LIGANDS FOR CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2008-08-07 WO disclosed