SCHEMBL4435170

SCHEMBL4435170

Cc1cccc(-c2cccc(S(N)(=O)=O)c2)c1C

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.55
CA1 P00915 8/20 0.55
CA9 Q16790 8/20 0.55
CA12 O43570 7/20 0.55
BRD4 O60885 1/20 0.50
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
CA4 P22748 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA13 Q8N1Q1 1/20 0.45
CREBBP Q92793 1/20 0.45
IKBKB O14920 2/20 0.45
CHUK O15111 1/20 0.45
TDO2 P48775 1/20 0.45
LRRK2 Q5S007 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL962658 0.88 CA1 (0.67) CA2CA1CA9CA12BRD4
SCHEMBL4073858 0.83 CA2 (0.74) CA2CA1CA9CA12CA4
SCHEMBL4733938 0.79 CA2 (0.64) CA2CA1CA9CA12BRD4
SCHEMBL15730257 0.78 IKBKB (0.52) CA2CA1CA9CA12BRD4
SCHEMBL16574040 0.76 CA2 (0.52) CA2CA1CA9CA12BRD4
SCHEMBL4135236 0.76 IKBKB (0.51) CA2CA1CA9CA12BRD4
SCHEMBL2308295 0.76 CA2 (0.56) CA2CA1CA9CA12BRD4
SCHEMBL28032548 0.76 CA2 (0.73) CA2CA1CA9CA12CA4
SCHEMBL30494473 0.75 PTGES2 (0.68) CA2CA1CA9CA12BRD4
SCHEMBL26462963 0.75 PTGES2 (0.68) CA2CA1CA9CA12BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884068-A 1- cyano-pyrolidin derivative as DUB inhibitor 特殊治疗有限公司 2018-11-23 CN disclosed
EP-2121621-A1 LXR AND FXR MODULATORS Exelixis, Inc. (US) 2009-11-25 EP disclosed
WO-2008073825-A1 LXR AND FXR MODULATORS EXELIXIS, INC. (US) 2008-06-19 WO disclosed