SCHEMBL4435568

SCHEMBL4435568

COc1ccc(C(CCN)c2ccc(C(F)(F)F)nc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
ALDH1A1 P00352 2/20 0.43
CYP19A1 P11511 1/20 0.41
HTT P42858 3/20 0.39
MITF O75030 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
P2RX7 Q99572 4/20 0.38
MAPK1 P28482 2/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
GPR35 Q9HC97 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
XBP1 P17861 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
BACE1 P56817 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
HRH1 P35367 1/20 0.37
SLC6A2 P23975 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4430222 0.81 FFAR1 (0.44) KMT2AMEN1ALDH1A1HTTLMNA
SCHEMBL4433142 0.80 SLC6A2 (0.55) KMT2AMEN1ALDH1A1HTTLMNA
SCHEMBL5947827 0.80 KMT2A (0.65) KMT2AMEN1ALDH1A1CYP19A1HTT
Hydrochloric Acid SCHEMBL4441383 0.79 SLC6A2 (0.54) KMT2AMEN1ALDH1A1HTTLMNA
SCHEMBL3736074 0.77 CYP1A2 (0.44) KMT2AMEN1ALDH1A1HTTMAPT
SCHEMBL4440597 0.76 SLC6A2 (0.42) KMT2AMEN1CYP19A1MAPTBACE1
SCHEMBL4435726 0.75 KMT2A (0.61) KMT2AMEN1ALDH1A1CYP19A1HTT
SCHEMBL10973267 0.75 HRH1 (0.67) KMT2AMEN1ALDH1A1HTTMITF
SCHEMBL4441702 0.73 CNR1 (0.48) KMT2AMEN1ALDH1A1HTTMITF
SCHEMBL4433971 0.73 CNR1 (0.48) KMT2AMEN1ALDH1A1HTTMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed