SCHEMBL4435792

SCHEMBL4435792

CN1CCc2cc(OC(=O)O)ccc2C1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 7/20 0.58
DRD5 P21918 6/20 0.58
DRD2 P14416 5/20 0.50
DRD3 P35462 5/20 0.50
HRH3 Q9Y5N1 1/20 0.50
DRD4 P21917 3/20 0.49
MAOA P21397 3/20 0.47
MAOB P27338 3/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
SLC6A4 P31645 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
AKR1C3 P42330 1/20 0.44
F10 P00742 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4438820 0.98 DRD1 (0.57) DRD1DRD5DRD2DRD3HRH3
SCHEMBL4057707 0.95 DRD1 (0.52) DRD1DRD5DRD2DRD3HRH3
Hydrochloric Acid SCHEMBL4563201 0.94 DRD1 (0.53) DRD1DRD5DRD2DRD3HRH3
SCHEMBL4563167 0.87 DRD1 (0.42) DRD1DRD5DRD2DRD3HRH3
SCHEMBL7286091 0.82 HRH3 (0.56) DRD1DRD5DRD2DRD3HRH3
SCHEMBL18034987 0.81 DRD1 (0.61) DRD1DRD5DRD2DRD3HRH3
SCHEMBL20119176 0.81 DRD1 (0.51) DRD1DRD5DRD2DRD3HRH3
SCHEMBL14340583 0.79 DRD1 (0.88) DRD1DRD5DRD2DRD3DRD4
SCHEMBL29515933 0.79 DRD1 (0.88) DRD1DRD5DRD2DRD3DRD4
SCHEMBL875632 0.79 ALOX15 (0.57) HRH3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-B1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2012-10-24 EP disclosed
EP-2132193-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS Boehringer Ingelheim International GmbH (DE) 2009-12-16 EP disclosed
WO-2008116881-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-02 WO disclosed
EP-1975165-A1 Substituted pyrrolidinamides, their production and utilisation as medicine Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2008-10-01 EP disclosed