SCHEMBL4057707

SCHEMBL4057707

CN1CCc2ccc(OC(=O)O)cc2C1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.52
DRD5 P21918 5/20 0.52
HRH3 Q9Y5N1 2/20 0.48
DRD2 P14416 4/20 0.47
DRD3 P35462 4/20 0.47
DRD4 P21917 2/20 0.47
MAOA P21397 4/20 0.46
MAOB P27338 4/20 0.46
SLC6A4 P31645 1/20 0.46
AKR1C3 P42330 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4435792 0.95 DRD1 (0.58) DRD1DRD5HRH3DRD2DRD3
Hydrochloric Acid SCHEMBL4438820 0.94 DRD1 (0.57) DRD1DRD5HRH3DRD2DRD3
Hydrochloric Acid SCHEMBL4563201 0.92 DRD1 (0.53) DRD1DRD5HRH3DRD2DRD3
SCHEMBL4563167 0.89 DRD1 (0.42) DRD1DRD5HRH3DRD2DRD3
SCHEMBL7286091 0.80 HRH3 (0.56) DRD1DRD5HRH3DRD2DRD3
SCHEMBL3723319 0.78 NR1H2 (0.67) HRH3
SCHEMBL29843474 0.78 DRD1 (0.79) DRD1DRD5DRD2DRD3DRD4
SCHEMBL4317508 0.78 DRD1 (0.79) DRD1DRD5DRD2DRD3DRD4
SCHEMBL20119176 0.76 DRD1 (0.51) DRD1DRD5HRH3DRD2DRD3
SCHEMBL875632 0.76 ALOX15 (0.57) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed