SCHEMBL4436230

SCHEMBL4436230

COc1ccccc1C(=NO)NO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.47
HDAC8 Q9BY41 1/20 0.45
HDAC1 Q13547 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
STAT3 P40763 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 2/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
KCNK3 O14649 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21163688 0.81 CTSD (0.47) CTSDGAAMAPTTSHRMAPK1
SCHEMBL17133942 0.75 CA1 (0.48) CTSDMAPTTSHRSTAT3NPC1
SCHEMBL17133940 0.75 CA1 (0.48) CTSDMAPTTSHRSTAT3NPC1
SCHEMBL2120412 0.73 CA1 (0.46) CTSDMAPTTSHRSTAT3NPC1
SCHEMBL470307 0.73 CA1 (0.46) CTSDMAPTTSHRSTAT3NPC1
SCHEMBL23879961 0.73 GAA (0.61) CTSDGAAMAPTTSHRSTAT3
SCHEMBL30210823 0.73 CA1 (0.46) CTSDMAPTTSHRSTAT3NPC1
SCHEMBL2775341 0.73 LMNA (0.51) CTSDHDAC8HDAC1GAASTAT3
SCHEMBL6671288 0.73 CTSD (0.70) CTSDGAAMAPTTSHRMAPK1
SCHEMBL105256 0.73 GAA (0.61) CTSDGAAMAPTTSHRSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125797-A1 AMINO- PYRIDINE DERIVATIVES AS S1P1 /EDG1 RECEPTOR AGONISTS Actelion Pharmaceuticals Ltd. (CH) 2009-12-02 EP disclosed
WO-2008114157-A1 AMINO- PYRIDINE DERIVATIVES AS S1P1 /EDG1 RECEPTOR AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2008-09-25 WO disclosed