SCHEMBL4438971

SCHEMBL4438971

CCCc1nc(Nc2ccc(C(=O)Nc3cc(CN(C)Cc4ccccc4)ccc3C)cc2)nc2ccccc12

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.43
ABL1 P00519 1/20 0.42
CTNNB1 P35222 4/20 0.40
TCF7L2 Q9NQB0 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4130118 0.93 MEN1 (0.45) HDAC1ABL1CTNNB1TCF7L2MEN1
SCHEMBL4132964 0.89 HDAC1 (0.46) HDAC1ABL1CTNNB1TCF7L2MEN1
SCHEMBL4138326 0.87 HDAC1 (0.48) HDAC1ABL1CTNNB1TCF7L2MAPT
SCHEMBL4130124 0.86 HDAC1 (0.44) HDAC1ABL1CTNNB1TCF7L2MAPT
SCHEMBL4138442 0.83 HDAC1 (0.49) HDAC1ABL1CTNNB1TCF7L2MAPT
SCHEMBL4449009 0.83 ABL1 (0.46) HDAC1ABL1CTNNB1TCF7L2MAPT
SCHEMBL4449995 0.82 SMN1; SMN2 (0.47) HDAC1ABL1KMT2AMAPT
SCHEMBL27781589 0.80 HDAC1 (0.51) HDAC1MEN1KMT2AMAPT
SCHEMBL4129999 0.80 HDAC1 (0.48) HDAC1ABL1CTNNB1TCF7L2MAPT
SCHEMBL4132202 0.80 BACE1 (0.47) HDAC1ABL1CTNNB1TCF7L2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134695-A1 INHIBITORS OF THE HEDGEHOG PATHWAY Exelixis, Inc. (US) 2009-12-23 EP disclosed
WO-2008112913-A1 INHIBITORS OF THE HEDGEHOG PATHWAY EXELIXIS, INC. (US) 2008-09-18 WO disclosed