SCHEMBL4449995

SCHEMBL4449995

CCCc1nc(Nc2ccc(C(=O)Nc3cc(CN4CCOCC4)ccc3C)cc2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
MAPT P10636 3/20 0.47
LMNA P02545 3/20 0.47
MAPK1 P28482 3/20 0.47
GALR3 O60755 1/20 0.47
RAB9A P51151 5/20 0.47
NPC1 O15118 2/20 0.47
KMT2A Q03164 1/20 0.47
HIF1A Q16665 3/20 0.47
EPAS1 Q99814 3/20 0.47
BCHE P06276 1/20 0.46
ABL1 P00519 1/20 0.45
BCR P11274 1/20 0.45
HDAC1 Q13547 1/20 0.45
TSHR P16473 1/20 0.45
STAT3 P40763 1/20 0.45
CDK2 P24941 2/20 0.44
FLT3 P36888 1/20 0.44
CCNA1 P78396 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4142803 0.94 MAPT (0.49) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4147051 0.90 HIF1A (0.51) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4151375 0.88 LRRK2 (0.59) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4139081 0.88 HDAC1 (0.50) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4134801 0.87 MAPT (0.48) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4144454 0.86 SMN1; SMN2 (0.47) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4137724 0.84 NPC1 (0.50) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL27963367 0.83 SMN1; SMN2 (0.44) SMN1; SMN2MAPTLMNAMAPK1GALR3
SCHEMBL4438971 0.82 HDAC1 (0.43) MAPTKMT2AABL1HDAC1
SCHEMBL27955756 0.81 LMNA (0.49) SMN1; SMN2MAPTLMNAMAPK1GALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134695-A1 INHIBITORS OF THE HEDGEHOG PATHWAY Exelixis, Inc. (US) 2009-12-23 EP disclosed
WO-2008112913-A1 INHIBITORS OF THE HEDGEHOG PATHWAY EXELIXIS, INC. (US) 2008-09-18 WO disclosed