SCHEMBL4444718

SCHEMBL4444718

COc1cc(COc2ccc(C=O)cc2)c2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.48
NPC1 O15118 3/20 0.47
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 3/20 0.46
OPRL1 P41146 1/20 0.45
ADAM17 P78536 3/20 0.44
MMP13 P45452 1/20 0.44
LMNA P02545 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PKM P14618 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7252416 0.87 NPC1 (0.48) RAB9ANPC1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL4058393 0.85 ADAM17 (0.60) OPRL1ADAM17MMP13
SCHEMBL6633312 0.82 GPBAR1 (0.53) RAB9ANPC1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5220040 0.81 NPC1 (0.44) RAB9ANPC1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL9582777 0.76 ALDH1A1 (0.56) RAB9ANPC1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL19422787 0.75 NPC1 (0.49) NPC1ALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL7069563 0.74 PPARA (0.60)
SCHEMBL3968933 0.73 POLB (0.47) NPC1ALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL3967858 0.73 ADAM17 (0.58) ADAM17MMP13
SCHEMBL15009057 0.73 ALDH1A1 (0.57) RAB9ANPC1ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397137-B1 HYDANTION DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES BRISTOL MYERS SQUIBB CO (US) 2009-10-14 EP disclosed