SCHEMBL4445394

SCHEMBL4445394

CC(=O)Nc1cccc2c(S(=O)(=O)NC(C)c3ccccc3)cccc12

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
KMT2A Q03164 1/20 0.50
EDNRA P25101 1/20 0.50
USP30 Q70CQ3 5/20 0.49
GFER P55789 1/20 0.45
RAB9A P51151 2/20 0.44
LMNA P02545 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14919627 0.85 ALDH1A1 (0.53) POLBLMNA
SCHEMBL4445405 0.84 EDNRA (0.47) POLBKMT2AEDNRAUSP30
SCHEMBL4450870 0.83 EDNRA (0.48) KMT2AEDNRAUSP30
SCHEMBL4446896 0.79 CCR8 (0.64) KMT2AEDNRAGFER
SCHEMBL6073751 0.78 EDNRA (0.58) POLBKMT2AEDNRALMNARXFP1
SCHEMBL24170513 0.78 CCR8 (0.66)
SCHEMBL30394968 0.78 CCR8 (0.66)
SCHEMBL4449277 0.78 NSD2 (0.56) EDNRA
SCHEMBL8054308 0.77 EDNRA (0.57) POLBKMT2AEDNRALMNARXFP1
SCHEMBL2372669 0.77 EDNRA (0.57) POLBKMT2AEDNRAUSP30LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547716-B2 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-06-16 US disclosed
EP-1402890-B1 SULFONAMIDE DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2008-01-09 EP disclosed
US-20040234622-A1 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2004-11-25 US disclosed
EP-1402890-A1 SULFONAMIDE DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2004-03-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040234622-A1 Sulfonamide derivatives PCNA, TOP2A, DDB1 POLB 56/4885KMT2A 460/4885EDNRA 1812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.