SCHEMBL4446276

SCHEMBL4446276

NC(=O)n1cnc2c(=O)[nH]c(N)nc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 6/20 0.54
TK1 P04183 2/20 0.53
PNP P00491 6/20 0.52
BLM P54132 2/20 0.52
USP2 O75604 1/20 0.52
TSHR P16473 1/20 0.52
EDNRA P25101 1/20 0.52
HTR2A P28223 1/20 0.52
RECQL P46063 1/20 0.52
HBB P68871 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
CYP3A4 P08684 1/20 0.50
NFKB1 P19838 1/20 0.50
VCP P55072 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HIF1A Q16665 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrimidine SCHEMBL27782384 0.91 XDH (0.49) XDHTK1PNPBLMUSP2
SCHEMBL27541246 0.89 XDH (0.58) XDHTK1PNPBLMUSP2
SCHEMBL27923065 0.89 XDH (0.55) XDHTK1PNPBLMUSP2
SCHEMBL2940017 0.86 XDH (0.52) XDHTK1PNPBLMUSP2
SCHEMBL218668 0.86 XDH (0.53) XDHTK1PNPBLMUSP2
SCHEMBL8029345 0.84 TK1 (0.48) XDHTK1PNPBLMUSP2
SCHEMBL4657411 0.84 TK1 (0.51) XDHTK1PNPBLMUSP2
SCHEMBL7765224 0.84 TK1 (0.57) XDHTK1PNPBLMUSP2
SCHEMBL1746164 0.83 TK1 (0.37) XDHTK1PNPBLMUSP2
SCHEMBL704009 0.82 XDH (0.50) XDHTK1PNPBLMUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040209352-A1 Integrated electrode and cell immobilization device equipped with the integrated electrode MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD (JP) 2004-10-21 US claimed
US-9914746-B2 Oligonucleotides containing high concentrations of guanine monomers KUROS BIOSCIENCES AG (CH) 2018-03-13 US disclosed
EP-2125854-B1 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS KUROS BIOSCIENCES AG (CH) 2016-10-26 EP disclosed
US-20160145293-A1 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS KUROS US LLC 2016-05-26 US disclosed
US-20140200338-A1 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS CYTOS BIOTECHNOLOGY AG (CH) 2014-07-17 US disclosed
US-8586728-B2 Oligonucleotides containing high concentrations of guanine monomers CYTOS BIOTECHNOLOGY AG (CH) 2013-11-19 US disclosed
CN-101611048-B Oligonucleotides containing high concentrations of guanine monomers CYTOS BIOTECHNOLOGY AG 2012-11-07 CN disclosed
CN-101611048-A The oligonucleotide that contains high concentrations of guanine monomers INTEGRATED DNA TECH INC (US) 2009-12-23 CN disclosed
EP-2125854-A2 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS Integrated DNA Technologies, Inc. (US) 2009-12-02 EP disclosed
WO-2008073960-A2 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS INTEGRATED DNA TECHNOLOGIES, INC. (US) 2008-06-19 WO disclosed
US-20080139797-A1 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS INTEGRATED DNA TECHNOLOGIES, INC. (US) 2008-06-12 US disclosed
US-20040209352-A1 Integrated electrode and cell immobilization device equipped with the integrated electrode MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD (JP) 2004-10-21 US disclosed
US-5952183-A CONCENTRATING AND PURIFYING ADDUCTS ISOLATED FROM BIOLOGICAL SOURCES USING IMMUNOAFFINITY CHROMATOGRAPHY BY COUPLING ANTI-ADDUCT ANTIBODIES TO SOLID MATRIX, APPLYING SAMPLE, WASHING MATRIX, ELUTING ADDUCTS PREVENTION LLC 1999-09-14 US disclosed
US-5840889-A POTENTIAL BIOMARKERS FOR DETERMINING SUSCEPTIBILITY OF ANIMALS TO A NUMBER OF ESTROGEN RELATED CANCERS THE BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 1998-11-24 US disclosed
WO-1997040061-A1 ESTROGEN-PURINE BASE, ESTROGEN-MERCAPTURATE ADDUCTS, AND FLUORESCENT PROBES AND MONOCLONAL ANTIBODIES THEREOF BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 1997-10-30 WO disclosed