SCHEMBL4447346

SCHEMBL4447346

COc1c(C(C)C)cc(C(=O)N[C@H](C(N)=O)C(c2ccccc2)c2ccccc2)cc1C(C)C

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
RXFP1 Q9HBX9 1/20 0.43
HPGDS O60760 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
CRHBP P24387 1/20 0.42
HTT P42858 1/20 0.42
CRHR2 Q13324 1/20 0.42
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 1/20 0.39
GPR139 Q6DWJ6 3/20 0.39
USP2 O75604 1/20 0.39
SLC1A2 P43004 1/20 0.38
PPARA Q07869 1/20 0.38
GLRA1 P23415 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447350 1.00 ALDH1A1 (0.46) ALDH1A1RXFP1HPGDSKDM4EMAPT
SCHEMBL4454641 0.87 ALDH1A1 (0.45) ALDH1A1RXFP1KDM4EMAPTCRHBP
SCHEMBL4454637 0.87 ALDH1A1 (0.45) ALDH1A1RXFP1KDM4EMAPTCRHBP
SCHEMBL14024227 0.86 RXFP1 (0.43) ALDH1A1RXFP1HPGDSHTTLMNA
SCHEMBL4446586 0.82 TNFRSF1A (0.46) ALDH1A1RXFP1HPGDSKDM4EMAPT
SCHEMBL4446583 0.82 TNFRSF1A (0.46) ALDH1A1RXFP1HPGDSKDM4EMAPT
SCHEMBL4450195 0.79 ALDH1A1 (0.54) ALDH1A1RXFP1MAPTGAAPKM
SCHEMBL4450186 0.79 ALDH1A1 (0.54) ALDH1A1RXFP1MAPTGAAPKM
SCHEMBL4448620 0.77 S1PR3 (0.47) ALDH1A1RXFP1MAPTHTTGAA
SCHEMBL4448626 0.77 S1PR3 (0.47) ALDH1A1RXFP1MAPTHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090012010-A1 Amino acid derivatives as calcium channel blockers NEUROMED PHRAMACEUTICALS LTD. (CA) 2009-01-08 US disclosed
US-20090012010-A1 Amino acid derivatives as calcium channel blockers NEUROMED PHRAMACEUTICALS LTD. (CA) 2009-01-08 US disclosed
US-20090012010-A1 Amino acid derivatives as calcium channel blockers NEUROMED PHRAMACEUTICALS LTD. (CA) 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012010-A1 Amino acid derivatives as calcium channel blockers CACNA1G, CACNA1H, CACNA1I ALDH1A1 2335/4885RXFP1 2511/4885HPGDS 1299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.