SCHEMBL4448481

SCHEMBL4448481

CC1(C)OCc2c(C(=O)NC3(c4ccc(F)cc4)CC3)cnc(C(=O)O)c2O1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.37
HDAC1 Q13547 4/20 0.37
HDAC2 Q92769 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
PTGER4 P35408 3/20 0.36
CCR1 P32246 2/20 0.35
ADRB1 P08588 1/20 0.35
KCNH2 Q12809 1/20 0.35
HSD17B13 Q7Z5P4 1/20 0.34
AKT1 P31749 4/20 0.33
CTSS P25774 2/20 0.33
PDE2A O00408 1/20 0.33
MAOB P27338 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12444452 0.91 HDAC3 (0.36) HDAC3HDAC1HDAC2HDAC6PTGER4
SCHEMBL12515762 0.91 HDAC3 (0.43) HDAC3HDAC1HDAC2HDAC6PTGER4
SCHEMBL15746733 0.82 ALDH1A1 (0.38) HDAC3HDAC1HDAC2HDAC6PTGER4
SCHEMBL15746653 0.77 KMT2A (0.40) MAOBMAPK1
SCHEMBL2216339 0.75 HDAC6 (0.44) HDAC3HDAC1HDAC2HDAC6MAOB
SCHEMBL12935668 0.74 KMT2A (0.42) MAOBMAPK1
SCHEMBL1503297 0.72 MAPT (0.43) MAPK1
SCHEMBL1503145 0.71 MAOB (0.37) MAOBMAPK1
SCHEMBL4316603 0.69 PTPN1 (0.38) MAPK1
SCHEMBL2146752 0.68 HSD11B1 (0.35) MAOBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO claimed