SCHEMBL4449174

SCHEMBL4449174

CC(C)(N)c1cccc(CCN)c1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 9/20 0.70
DRD2 P14416 1/20 0.50
DRD1 P21728 1/20 0.50
MAOB P27338 2/20 0.48
NOS1 P29475 1/20 0.46
KIF11 P52732 3/20 0.45
HTR2A P28223 2/20 0.45
CYP2A6 P11509 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.45
HTR7 P34969 1/20 0.45
HTR2C P28335 2/20 0.44
HTR6 P50406 2/20 0.44
HTR2B P41595 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911870 0.86 TAAR1 (0.67) TAAR1DRD2DRD1MAOBNOS1
Hydrochloric Acid SCHEMBL14157546 0.85 TAAR1 (0.65) TAAR1DRD2DRD1MAOBNOS1
SCHEMBL4454237 0.84 KIF11 (0.49) TAAR1MAOBNOS1KIF11HTR2A
SCHEMBL18434546 0.83 TAAR1 (0.73) TAAR1DRD2DRD1MAOBNOS1
SCHEMBL40017 0.82 TAAR1 (1.00) TAAR1DRD2DRD1MAOBHTR2A
SCHEMBL3177646 0.82 KIF11 (0.50) TAAR1KIF11HTR2AHTR2CHTR2B
SCHEMBL24351980 0.81 TAAR1 (0.61) TAAR1DRD2DRD1MAOBNOS1
Hydrochloric Acid SCHEMBL27033001 0.81 TAAR1 (0.71) TAAR1DRD2DRD1MAOBNOS1
Iodide SCHEMBL31174197 0.81 TAAR1 (0.96) TAAR1DRD2DRD1MAOBHTR2A
Methane SCHEMBL28404139 0.81 TAAR1 (0.96) TAAR1DRD2DRD1MAOBHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-0819000-A4 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2001-04-11 EP disclosed
US-5962499-A ACARICIDAL, ANTIPARASITIC, INSECTICIDAL AND ANTHELMINTIC AGENTS MERCK & CO., INC. (US) 1999-10-05 US disclosed
CN-1184423-A Nodulisporic acid derivatives MERCK & CO INC (US) 1998-06-10 CN disclosed
EP-0819000-A1 NODULISPORIC ACID DERIVATIVES Merck & Co., Inc. (US) 1998-01-21 EP disclosed
WO-1996029073-A1 NODULISPORIC ACID DERIVATIVES MERCK & CO., INC. (US) 1996-09-26 WO disclosed