SCHEMBL4449803

SCHEMBL4449803

COc1cc(N2CCN(C(C=O)n3nc(I)c(Cl)c3C)[C@@H](C)C2)c(F)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPOX P50336 2/20 0.36
CCR1 P32246 14/20 0.36
ROCK2 O75116 3/20 0.33
PRKG1 Q13976 3/20 0.33
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016337 0.87 CCR1 (0.37) PPOXCCR1ALDH1A1LMNATP53
SCHEMBL3469130 0.85 CCR1 (0.46) CCR1
SCHEMBL3638427 0.83 CCR1 (0.35) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL4013895 0.81 PPOX (0.34) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL3632434 0.79 PPOX (0.43) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL3726336 0.79 PPOX (0.43) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL4020093 0.79 CCR1 (0.43) CCR1
SCHEMBL3632485 0.77 PPOX (0.35) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL3640517 0.77 ROCK2 (0.38) PPOXCCR1ROCK2PRKG1ALDH1A1
SCHEMBL3633830 0.77 ROCK2 (0.39) PPOXROCK2PRKG1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed