SCHEMBL445483

SCHEMBL445483

CC(N)C(=O)C(N)(CSSCC(N)(C(=O)O)C(=O)C(C)N)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33
NOS3 P29474 1/20 0.32
GRM2 Q14416 1/20 0.32
GRM3 Q14832 1/20 0.32
GABRP O00591 2/20 0.30
GABRD O14764 2/20 0.30
GABRA1 P14867 2/20 0.30
GABRB1 P18505 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA5 P31644 2/20 0.30
GABRA3 P34903 2/20 0.30
GABRA2 P47869 2/20 0.30
GABRB2 P47870 2/20 0.30
GABRA4 P48169 2/20 0.30
GABRE P78334 2/20 0.30
GABRA6 Q16445 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9810240 1.00 SMN1; SMN2 (0.34) SMN1; SMN2HIF1ANOS1NOS2NOS3
SCHEMBL9326098 0.88 KIF11 (0.36) NOS1NOS2NOS3SLC7A5
SCHEMBL10422578 0.88 KIF11 (0.36) NOS1NOS2NOS3SLC7A5
SCHEMBL441158 0.84 ALOX15 (0.42)
SCHEMBL10421342 0.82 SLC7A5 (0.47) SMN1; SMN2HIF1AGRM2GRM3SLC7A5
SCHEMBL9810245 0.80 DPP4 (0.36)
SCHEMBL30863909 0.79 CYP1A2 (0.36) SMN1; SMN2HIF1AGRM2GRM3GABRP
SCHEMBL8475144 0.74
SCHEMBL27527294 0.74
SCHEMBL8820876 0.74 GRM2 (0.34) NOS1NOS2NOS3GRM2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110418837-B Culture medium comprising oligopeptides 赢创运营有限公司 2024-04-02 CN disclosed
EP-3372671-B1 CULTURE MEDIUM COMPRISING OLGOPEPTIDES EVONIK OPERATIONS GMBH (DE) 2021-11-03 EP disclosed
EP-1144613-B2 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY INC (US) 2020-05-06 EP disclosed
WO-2018162346-A1 CULTURE MEDIUM COMPRISING OLIGOPEPTIDES EVONIK TECHNOCHEMIE GMBH (DE) 2018-09-13 WO disclosed
EP-3372671-A1 CULTURE MEDIUM COMPRISING OLGOPEPTIDES Evonik Technochemie GmbH (DE) 2018-09-12 EP disclosed
US-20170362626-A1 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY, INC. 2017-12-21 US disclosed
US-20160244798-A1 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY, INC. 2016-08-25 US disclosed
EP-2305804-B1 MonoPEGylated human growth hormone BOLDER BIOTECHNOLOGY INC (US) 2015-05-06 EP disclosed
US-8957023-B2 Methods for making proteins containing free cysteine residues BOLDER BIOTECHNOLOGY INC. (US) 2015-02-17 US disclosed
US-8932828-B2 Method for preparing recombinant granulocyte colony stimulating factor cysteine muteins BOLDER BIOTECHNOLOGY, INC. (US) 2015-01-13 US disclosed
US-20040018586-A1 Lysis, denaturing, reducing Growth hormones NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-01-29 US disclosed
EP-1284987-A2 METHODS FOR REFOLDING PROTEINS CONTAINING FREE CYSTEINE RESIDUES Bolder Biotechnology, Inc. (US) 2003-02-26 EP disclosed
EP-1144613-A4 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY INC (US) 2002-10-29 EP disclosed
WO-2001087925-A2 METHODS FOR REFOLDING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY, INC. (US) 2001-11-22 WO disclosed
EP-1144613-A1 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES Bolder Biotechnology, Inc. (US) 2001-10-17 EP disclosed
WO-2000042175-A1 METHODS FOR MAKING PROTEINS CONTAINING FREE CYSTEINE RESIDUES BOLDER BIOTECHNOLOGY INC. (US) 2000-07-20 WO disclosed
EP-0264953-B1 USE OF N,N'-BIS-L-AMINO ACID-L-CYSTIN PEPTIDES IN AMINO ACID PREPARATIONS FOR ORAL AND PARENTERAL ADMINISTRATION PFRIMMER KABI GMBH & CO. KG (DE) 1991-05-08 EP disclosed
US-4968696-A CHRONIC UREMIA OR HEPATIC CIRRHOSIS PFRIMMER + CO. PHARMAZEUTISCHE WERKE ERLANGEN GMBH + CO. KG (DE) 1990-11-06 US disclosed
WO-1988003150-A2 N,N'-BIS-AMINO ACID-L-CYSTINE-PEPTIDE-CONTAINING AMINO ACID PREPARATIONS FOR ORAL AND PARENTERAL ADMINISTRATION PFRIMMER + CO. PHARMAZEUTISCHE WERKE ERLANGEN GMBH (DE) 1988-05-05 WO disclosed
EP-0264953-A2 Use of N,N'-bis-L-amino acid-L-cystin peptides in amino acid preparations for oral and parenteral administration PFRIMMER KABI GMBH & CO. KG (DE) 1988-04-27 EP disclosed