SCHEMBL4456586

SCHEMBL4456586

CCN(CC)CCN(CCO)C(=O)CCOCCc1cccc2ccccc12.O=C(Cl)C(=O)Cl

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.55
CDYL Q9Y232 1/20 0.53
KDM4E B2RXH2 3/20 0.50
HTR2A P28223 5/20 0.36
CYP3A4 P08684 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
DRD1 P21728 1/20 0.36
SLC6A4 P31645 1/20 0.36
OPRM1 P35372 1/20 0.36
DRD3 P35462 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180012 0.96 ADRB2 (0.58) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL1180543 0.84 ADRB2 (0.59) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL1179648 0.82 ADRB2 (0.53) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL12193241 0.82 ADRB2 (0.54) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL3577973 0.79 ADRB2 (0.54) ADRB2KDM4ECHRM2CHRM1DRD1
Oxalic Acid SCHEMBL6773522 0.76 KDM4E (0.72) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL3813478 0.76 CDYL (0.64) ADRB2CDYLKDM4EHTR2ACYP3A4
SCHEMBL29372244 0.72 ADRB2 (1.00) ADRB2
SCHEMBL186048 0.72 ADRB2 (1.00) ADRB2
SCHEMBL3587177 0.71 ADRB2 (0.44) ADRB2CDYLKDM4ECYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124941-A1 COMBINATION OF A MUSCARINIC RECEPTOR ANTAGONIST AND A BETA-2-ADRENOCEPTOR AGONIST Argenta Discovery Limited (GB) 2009-12-02 EP disclosed
WO-2008096126-A1 COMBINATION OF A MUSCARINIC RECEPTOR ANTAGONIST AND A BETA-2-ADRENOCEPTOR AGONIST ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed